beta-adrenergic-receptor kinase EC#: 2.7.11.15; ChemWhat Code: 1379019

Product Name beta-adrenergic-receptor kinase
Example Structure Example Structure of beta-adrenergic-receptor kinase EC#: 2.7.11.15
Synonyms ark, bARKct, beta adrenergic receptor kinase, beta-adrenergic receptor kinase, beta-adrenergic receptor kinase 1, beta-adrenergic receptor kinase 2, beta-adrenergic receptor-specific kinase, beta-AR kinase, beta-ARK, beta-ARK 1, beta-ARK 2, beta-receptor kinase, betaAR kinase 1, betaARK, betaARK1, betaARK2, betabeta-adrenergic receptor kinase 1, carboxyl-terminus of beta-adrenergic receptor kinase, G protein-coupled receptor kinase, G protein-coupled receptor kinase 2, G protein-coupled receptor kinase 3, G protein-coupled receptor kinase-2, G protein-coupled receptor kinase-3, G protein-coupled receptor regulatory kinase, G protein-coupled receptor regulatory kinase 2, G-protein coupled receptor kinase 2, G-protein receptor kinase 2, G-protein-coupled receptor kinase 2, G-protein-coupled receptor kinase-2, GPCR kinase, GPCR kinase 2, Gprk2, GRK, GRK2, GRK3, GRK5, guanine nucleotide-binding protein-coupled receptor kinase, kinase (phosphorylating), beta-adrenergic-receptor, More
EC Number 2.7.11.15
CAS Registry Number 102925-39-3
Comments Requires G-protein for activation and therefore belongs to the family of G-protein-dependent receptor kinases (GRKs). Acts on the agonist-occupied form of the receptor; also phosphorylates rhodopsin, but more slowly. Does not act on casein or histones. The enzyme is inhibited by Zn2+?and digitonin but is unaffected by cyclic-AMP (cf. EC?2.7.11.14, rhodopsin kinase and EC?2.7.11.16, G-protein-coupled receptor kinase).
Cofactor
History
Reactions Atp + [beta-adrenergic receptor] = adp + [beta-adrenergic receptor] phosphate.

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